Chemical & Pharmaceutical Structure Analysis

Where Technology and Solutions Meet...
Where East Meets West

CPSA Shanghai 2011

Changing Paradigm in Drug Discovery & Development:
East Meets West

April 13 - 16, 2011
Renaissance Shanghai Pudong Hotel
Shanghai, China


Abstract

Thursday PM - Parallel Session I

Predictive Toxicology Approaches for Small Molecule Oncology Drugs

Vic Kadambi
Millennium Pharmaceuticals, Cambridge, MA USA

A daunting, unmet medical need exists for effective oncology chemotherapies, with cancer deaths in 2009 to exceed 560,000 in the United States alone. Because of the rapid demise of the majority of cancer patients with metastatic disease, oncology drug development must follow a much different paradigm than therapeutic candidates for less onerous diseases. The majority of drug candidates in development today are targeted at cancer therapy. Many of these candidate chemotherapeutic agents are active against novel targets, often presenting unique toxicological profiles. Since many of these novel targets are not unique to cancer cells, therapeutic margins may not exist. Decision making, in this event, is among the most challenging that any pharmaceutical toxicologist/pathologist or regulator will face. Nonclinical development scientists must compress timelines to present therapeutic options for cancer patients who have failed conventional therapy. In support of this goal, the U. S. Food and Drug Administration has created an oncology-specific paradigm for nonclinical testing and has introduced strategies to accelerate development and approval of successful candidates. Pharmaceutical toxicology testing strategies must not only satisfy regulation as the minimal expectation, but also attempt to reduce the current high attrition rates for oncologic candidates. A successful toxicology testing strategy represents the substance of this treatise.




Dr. Vivek (Vic) Kadambi is the head of the Drug Safety & Evaluation Group at Millennium: The Takeda Oncology Company. Dr. Kadambi has a B.S. and a M.S. in Microbiology from the University of Bombay and a Ph.D. in Cardiovascular Pharmacology and Physiology from the University of Cincinnati. Dr. Kadambi was the recipient of the American Heart Association Fellowship, Ohio Affiliate (1997-1998) as well as the Young Investigator Award from the Heart Failure Society of America (1998). In addition, he was awarded the Outstanding Contributor Award from Millennium Pharmaceuticals Inc (2001 and 2004). Dr. Kadambi has served as the Program Chair for pharmacology and toxicology related symposia and was a councilor for the New England Society of Toxicology (2004-2005). Dr. Kadambi represents Millennium on the Preclinical Safety Leadership Group of the International Consortium for Innovation and Quality in Pharmaceutical Development (IQ). Dr. Kadambi has presented several abstracts at both national as well as international meetings as well as published over peer reviewed manuscripts and 6 book chapters.

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